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Bepotastine Besilate
CAS No. 190786-44-8
Bepotastine Besilate ( Bepotastine besilate; TAU-284 )
Catalog No. M12990 CAS No. 190786-44-8
Bepotastine is a non-sedating, selective antagonist of histamine 1 (H1) receptor with pIC50 of 5.7.
Purity : >98%(HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 10MG | 35 | In Stock |
|
| 25MG | 63 | In Stock |
|
| 50MG | 110 | In Stock |
|
| 100MG | 165 | In Stock |
|
| 500MG | 413 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameBepotastine Besilate
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NoteResearch use only, not for human use.
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Brief DescriptionBepotastine is a non-sedating, selective antagonist of histamine 1 (H1) receptor with pIC50 of 5.7.
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DescriptionBepotastine is a non-sedating, selective antagonist of histamine 1 (H1) receptor with pIC50 of 5.7.
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SynonymsBepotastine besilate; TAU-284
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PathwayGPCR/G Protein
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TargetHistamine Receptor
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RecptorH1 receptor
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Research AreaInflammation/Immunology
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Indication——
Chemical Information
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CAS Number190786-44-8
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Formula Weight547.06
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Molecular FormulaC21H25ClN2O3·C6H6O3S
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Purity>98%(HPLC)
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SolubilityDMSO:109 mg/mL (199.24 mM); Ethanol:<1 mg/mL (<1 mM); Water:<1 mg/mL (<1 mM)
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SMILESC1CN(CCC1O[C@@H](C2=CC=C(C=C2)Cl)C3=CC=CC=N3)CCCC(=O)O.C1=CC=C(C=C1)S(=O)(=O)O
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Da Prada M, et al. J Pharmacol Exp Ther, 1989, 248(1), 400-414.
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